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N-(2-Chloro-4-hydroxyphenyl)-N'-cyclopropyl-urea CAS:796848-79-8
N-(2-Chloro-4-hydroxyphenyl)-N'-cyclopropyl-urea wani sinadari ne mai sinadaran da ke dauke da tsarin kwayoyin halitta C10H11ClN2O2. Yana cikin nau'in sinadaran urea da aka maye gurbinsu da rukunin chloro-hydroxyphenyl da rukunin cyclopropyl. An san wannan sinadari saboda sarkakiyar tsarinsa da kuma yuwuwar amfani da shi a cikin nazarin sinadarai da halittu daban-daban.
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1,4-Dihydro-7-methoxy-4-oxo-6-quinolinecarboxylic acid methyl ester CAS:205448-65-3
1,4-Dihydro-7-methoxy-4-oxo-6-quinolinecarboxylic acid methyl ester wani sinadari ne mai dauke da kwayoyin halitta C12H11NO4. Yana cikin rukunin quinoline na mahadi kuma ana siffanta shi da rukunin methyl ester da aka makala a zoben quinoline, tare da maye gurbin methoxy a matsayi na 7 da kuma rukunin keto a matsayi na 4.
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AZD-9291 mesylate CAS:1421373-66-1
AZD-9291 mesylate wani sinadari ne na magunguna wanda ke ɗauke da dabarar kwayoyin halitta C28H33N7O4∙CH4O3S. Yana cikin ajin masu hana tyrosine kinase kuma ana amfani da shi musamman wajen magance cutar kansar huhu ta ƙwayoyin halitta (NSCLC). Wannan maganin yana nufin kuma yana hana nau'ikan masu karɓar haɓakar epidermal growth factor (EGFR) da aka canza, waɗanda galibi ake samu a cikin ciwon daji na NSCLC.
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5-Chloromethyl-2H-1,2,4-triazolin-3-one CAS:252742-72-6
5-Chloromethyl-2H-1,2,4-triazolin-3-one wani muhimmin sinadari ne mai amfani da yawa a fannin ilmin sinadarai na likitanci da binciken agrochemical. Yana cikin rukunin abubuwan da aka samo daga triazolinone, wanda aka bambanta shi da wani tsari na musamman na kwayoyin halitta wanda ke ba da gudummawa ga ayyukan halittu da yuwuwar amfani da shi wajen warkar da cututtuka.
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5-CHLOROTHIOPHEN-2-CARBONYL CHLORIDE CAS:42518-98-9
5-Chlorothiophene-2-carbonyl chloride wani sinadari ne na sinadarai wanda ya samo asali daga ajin thienylacyl chlorides. An siffanta shi da tsarin kwayoyin halitta wanda ya kunshi zoben thiophene da aka maye gurbinsa da rukunin chloro a matsayi na 5 da kuma rukunin carbonyl chloride a matsayi na 2. Wannan sinadari yana da matukar sha'awa ga hadakar kwayoyin halitta saboda yawan amsawar sa da kuma yuwuwar amfani da shi a fannin magunguna da kimiyyar kayan aiki.
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5,6-Dihydro-3-(4-morpholinyl)-1-(4-nitrophenyl)-2(1H)-pyridinone CAS:503615-03-0
5,6-Dihydro-3-(4-morpholinyl)-1-(4-nitrophenyl)-2(1H)-pyridinone wani sinadari ne da aka sani da shi saboda tsarin kwayoyin halitta mai rikitarwa da kuma aikace-aikace daban-daban a fannin ilmin sinadarai na likitanci da binciken magunguna. Wannan sinadari yana cikin ajin pyridinones kuma an bambanta shi da tsarinsa na musamman na ƙungiyoyin aiki, waɗanda ke ba da takamaiman halaye masu mahimmanci ga ayyukansa na halitta.
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4-Chloro-2-methylsulfanyl-pyrimidine-5-carboxylic acid ethyl ester CAS:5909-24-0
4-Chloro-2-methylsulfanyl-pyrimidine-5-carboxylic acid ethyl ester wani sinadari ne da aka sani da muhimmiyar rawar da yake takawa a fannin ilmin sinadarai na likitanci da binciken magunguna. Kasancewarsa na cikin rukunin abubuwan da suka samo asali daga pyrimidine, wannan sinadari yana nuna wani tsari na musamman na kwayoyin halitta wanda yake da matukar muhimmanci ga ayyukansa na halitta da kuma aikace-aikacensa na warkewa.
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3-CHLORO-4-METHOXYBENZYLAMINE HYDROCHLORIDE CAS:41965-95-1
3-Chloro-4-Methoxybenzylamine Hydrochloride sanannen sinadari ne da aka san shi da shi sosai saboda aikace-aikacensa a fannin kimiyyar magunguna da binciken magunguna. Wannan sinadari yana cikin rukunin amines masu ƙamshi kuma an bambanta shi da takamaiman tsarinsa na ƙungiyoyin aiki masu mahimmanci ga ayyukansa na halitta.
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3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridina-2(1H)-daya CAS:545445-44-1
3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one wani sinadari ne da aka san shi da tsarin kwayoyin halitta mai rikitarwa da kuma aikace-aikace daban-daban a fannin ilmin sinadarai da ci gaban magunguna. Wannan sinadari yana cikin rukunin dihydropyridinones kuma an san shi da tsarinsa mai rikitarwa na ƙungiyoyi masu aiki, waɗanda ke ba da takamaiman halaye masu mahimmanci ga ayyukansa na halitta.
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L(-)-Thiazolidine-4-carboxylic acid CAS:34592-47-7
L(-)-Thiazolidine-4-carboxylic acid sanannen sinadari ne da aka san shi da amfaninsa daban-daban a fannin kimiyyar sinadarai da binciken magunguna. Kasancewarsa daga cikin nau'in thiazolidine, wannan sinadari yana da wani tsari na musamman na kwayoyin halitta don ayyukansa na halitta da kuma damar warkewa.
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Nintedanib CAS:656247-17-5
Nintedanib wani ƙaramin ƙwayar cuta ce mai ƙarfi wadda ke hana tyrosine kinase inhibitor (TKI) wanda ke da matuƙar muhimmanci a fannin maganin kansar da cututtukan fibrotic. Yana yin tasirinsa a fannin magunguna ta hanyar niyya ga ƙwayoyin tyrosine masu karɓar ƙwayoyin cuta da yawa waɗanda ke da hannu a cikin angiogenesis, fibrogenesis, da kuma daidaita ci gaban ƙari.
