Bel da Hanya: Haɗin gwiwa, Jituwa da Cin Nasara
samfurori

Kayayyaki

Letrozole CAS:112809-51-5 Mai Kaya na Masana'anta

Letrozole wani ɓangare ne na sabon ƙarni na masu hana aromatase masu zaɓe kuma wani nau'in benzotriazole ne da aka haɗa ta hanyar roba. Letrozole yana hana aromatase don rage matakan estrogen, don haka yana hana estrogen daga haɓaka ci gaban ƙari. Ayyukansa a cikin jiki ya fi ƙarfi sau 150-250 fiye da na Amarante na ƙarni na farko. Ganin cewa yana da zaɓi sosai, ba zai shafi aikin glucocorticoid, mineralocorticoid da thyroid ba; ko da a cikin allurai masu yawa, ba zai sami wani tasiri mai hana fitar da corticosteroid na adrenal ba, wanda hakan ke ba shi babban ma'aunin magani.


Cikakken Bayani game da Samfurin

Alamun Samfura

Aikace-aikace da Tasiri

Ana iya haɗa Letrazole a matakai biyu daga 4-bromomethyl-benzonitrile tare da 1,2,4-triazole kuma shine mai hana aromatase na ƙarni na uku. Yana da takamaiman hana P450arom wanda ke hana canza androstenedione zuwa estrone. Rage estrogen na plasma ya kasance nan take kuma yana ɗorewa. Ana cimma wannan ba tare da hana wasu steroid biosynthesis ba, wanda hakan ya sa ya zama mafi kyawun mai hana aromatase da aka gwada. Letrazole yana da aikin hana ƙari mai ban mamaki, yana da juriya sosai kuma ba shi da illa mai guba. Ya fi ƙarfin aminoglutethimide sau 10,000, a cikin jiki, farkon mai hana aromatase da aka kafa sosai.

Samfurin Samfuri

图片290(1)
图片222(1)

Shirya Samfurin:

shafi na 198 (1)

Ƙarin Bayani:

Tsarin aiki C17H11N5
Gwaji 99%
Bayyanar Foda fari
Lambar CAS 112809-51-5
shiryawa 25KG
Rayuwar shiryayye Shekaru 2
Ajiya A adana a wuri mai sanyi da bushewa
Takardar shaida ISO.

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