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tert-butyl 4-hydroxy-3,4-dihydroquinoline-1(2H)-carboxylate CAS: 932398-74-8
Tert-butyl 4-hydroxy-3,4-dihydroquinoline-1(2H)-carboxylate, wanda aka fi sani da compound Y, wani sinadari ne mai amfani da sinadarai masu yawa wanda ke da amfani mai yawa a masana'antun magunguna da kimiyyar kayan aiki. Tare da dabarar kwayoyin halitta ta C15H21NO3, wannan sinadari yana da wani sifa na quinoline na musamman wanda aka maye gurbinsa da ƙungiyar tert-butyl da aikin carboxylate. Tsarinsa na musamman yana ba da kyawawan halaye masu mahimmanci ga aikace-aikace daban-daban, tun daga haɗa magunguna zuwa sunadarai na kayan aiki. A matsayin babban matsakaici a cikin haɗa kwayoyin halitta, yana aiki a matsayin tushe don haɓaka sabbin magunguna da kayan aiki, yana haifar da ƙirƙira a sassa daban-daban.
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Semaglutide CAS:910463-68-2
Semaglutide wani agonist ne mai ƙarfi na glucagon-like peptide-1 (GLP-1) wanda ake amfani da shi wajen magance ciwon suga na nau'in 2 da kiba. Semaglutide, wanda yake kama da hormone na GLP-1 na ciki, yana ba da aikin magani na dogon lokaci saboda sauye-sauyen da yake yi tare da sarkar gefen fatty acid. Tare da dabarar kwayoyin halitta ta C187H291N45O59, tsawon rabin rayuwar semaglutide yana ba da damar yin allura sau ɗaya a mako, yana ƙara jin daɗin marasa lafiya da bin tsarin magani.
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Linaclotide CAS:851199-59-2
Linaclotide wani maganin guanylate cyclase-C (GC-C) ne da ake amfani da shi don magance maƙarƙashiya mai ɗorewa da kuma ciwon hanji mai saurin kamuwa da maƙarƙashiya (IBS-C). Linaclotide, wanda yake kama da peptide na guanylin na ciki, yana ɗaurewa da kuma kunna masu karɓar GC-C a cikin tsarin narkewar abinci, wanda ke haifar da ƙaruwar fitar ruwa daga hanji da kuma hanzarta lokacin wucewa. Tare da dabarar kwayoyin halitta ta C59H79N15O21S6, linaclotide tana ba da hanyar da aka yi niyya don rage maƙarƙashiya da rage rashin jin daɗin ciki da ke da alaƙa da IBS-C, yana inganta rayuwar marasa lafiya.
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Liraglutide CAS:204656-20-2
Liraglutide wani sinadari ne mai ƙarfi na glucagon-like peptide-1 (GLP-1) wanda ake amfani da shi wajen magance ciwon suga na nau'in 2 da kiba. Liraglutide, wanda yake kama da hormone na GLP-1 na ciki, yana ba da aikin magani na dogon lokaci saboda sauye-sauyen da yake yi tare da sarkar gefen fatty acid. Tare da dabarar kwayoyin halitta ta C172H265N43O51, tsawon rabin rayuwar liraglutide yana ba da damar shan magani sau ɗaya a rana, yana ƙara jin daɗin marasa lafiya da bin tsarin magani.
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ethyl 4-(hydroxymethyl)-1H-pyrazole-5-carboxylate CAS:61453-49-4
Ethyl 4-(hydroxymethyl)-1H-pyrazole-5-carboxylate, wani sinadari mai amfani da sinadarai, yana da mahimmanci a fannoni daban-daban na magunguna da sinadarai na noma. Tare da dabarar kwayoyin halitta C8H10N2O3, yana da zoben pyrazole wanda aka maye gurbinsa da rukunin ethyl, wani sinadari na hydroxymethyl, da kuma aikin carboxylate. Wannan sinadari yana aiki a matsayin matsakaici mai mahimmanci a cikin hadakar kwayoyin halitta, yana sauƙaƙa haɓaka nau'ikan magunguna da sinadarai na noma. Tsarinsa na musamman da ƙungiyoyin aiki sun sa ya zama tubalin gini mai amfani don haɗa ƙwayoyin halitta tare da aikace-aikace daban-daban, suna haifar da ƙirƙira a masana'antu da yawa.
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Ethyl 4-cyanopiperidine-4-carboxylatehydrochloride CAS:123730-64-3
Ethyl 4-cyanopiperidine-4-carboxylate hydrochloride, wani muhimmin sinadari ne na sinadarai, yana da tasiri a masana'antar magunguna da sinadarai na noma. Tare da dabarar kwayoyin halitta C9H14ClNO2, yana da zoben piperidine wanda aka maye gurbinsa da rukunin ethyl da kuma wani yanki na cyano, tare da aikin carboxylate, duk an haɗa shi da ion chloride. Wannan sinadari yana aiki a matsayin matsakaici mai mahimmanci a cikin haɗakar kwayoyin halitta, yana sauƙaƙa haɓaka nau'ikan magunguna da sinadarai na noma. Tsarinsa na musamman da ƙungiyoyin aiki sun sa ya zama tubalin gini mai amfani don haɗa ƙwayoyin halitta tare da aikace-aikace daban-daban, suna haɓaka ƙirƙira a fannoni da yawa.
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methyl imidazo[1,5-a]pyridine-7-carboxylate CAS:1377829-50-9
Methyl imidazo[1,5-a]pyridine-7-carboxylate, wani sinadari mai sinadarai tare da dabarar kwayoyin halitta C9H7N3O2, ya shahara saboda aikace-aikacensa masu yawa a fannin kimiyyar magunguna da kayan aiki. Tare da tsarin imidazo-pyridine, yana gabatar da halaye na musamman na tsarin da ke ba da gudummawa ga amfaninsa daban-daban. Wannan sinadari yana aiki a matsayin matsakaici mai mahimmanci a cikin hadakar kwayoyin halitta, yana aiki a matsayin tushe don haɓaka magunguna da kayan aiki. Tsarinsa na musamman da amsawarsa sun sa ya zama muhimmin sashi a cikin bincike da ayyukan masana'antu daban-daban, suna haifar da kirkire-kirkire a fannoni daban-daban.
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Arg34GLP-1 CAS:1169630-82-3
Arg34GLP-1, wanda kuma aka sani da Arginine-34 Glucagon-Like Peptide 1, wani sinadari ne mai aiki da sinadarai masu aiki wanda ke da tasiri mai mahimmanci a cikin daidaita metabolism da kuma hanyoyin magance ciwon suga da kiba. Wannan sinadari ya samo asali ne daga sinadarin glucagon-like peptide 1 (GLP-1) kuma yana da ragowar arginine a matsayi na 34. Tsarin kwayoyin halittarsa da ayyukansa na halitta sun sa ya zama ɗan takara mai kyau ga aikace-aikacen magunguna da nufin inganta yanayin glucose da haɓaka rage nauyi.
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1-tert-Butyl 4-ethyl 4-cyanopiperidine-1,4-dicarboxylate CAS:1016258-66-4
1-tert-Butyl 4-ethyl 4-cyanopiperidine-1,4-dicarboxylate wani sinadari ne da aka sani da amfaninsa daban-daban a masana'antun magunguna da sinadarai na noma. Tare da tsarin kwayoyin halitta C15H24N2O4, yana nuna tsarin tsari na musamman wanda ke nuna zoben piperidine wanda aka maye gurbinsa da ƙungiyoyin tert-butyl, ethyl, da cyano. Wannan sinadari yana aiki a matsayin matsakaici mai mahimmanci a cikin haɗakar kwayoyin halitta, yana taka muhimmiyar rawa wajen haɓaka magunguna daban-daban da sinadarai na noma. Tsarin maye gurbin dabarunsa da ƙungiyoyin aiki sun sa ya zama tubalin gini mai amfani don haɗa gine-ginen kwayoyin halitta masu rikitarwa tare da kyawawan halaye don aikace-aikace daban-daban.
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6-Chloro-3,4-dihydro-2H-benzo[b][1,4]oxazine hydrochloride CAS:1956310-17-0
6-Chloro-3,4-dihydro-2H-benzo[b][1,4]oxazine hydrochloride, wanda aka fi sani da compound X, wani sinadari ne mai amfani da dama a masana'antun magunguna da kimiyyar kayan aiki. Tare da dabarar kwayoyin halitta ta C8H8ClNO•HCl, wannan sinadari yana da wani sifa na benzo[b][1,4]oxazine wanda aka maye gurbinsa da kwayar chlorine. Tsarinsa na musamman ya sa ya zama matsakaici mai mahimmanci a cikin hadadden kwayoyin halitta, yana aiki a matsayin tushe don haɓaka magunguna daban-daban da kayan aiki masu aiki.
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8-Methylquinazolin-4(3H)-one CAS:19181-54-5
8-Methylquinazolin-4(3H)-one wani sinadari ne mai amfani da dama a fannin ilmin sinadarai na likitanci da kuma binciken magunguna. Tare da tsarin kwayoyin halittarsa na C9H8N2O, yana cikin rukunin sinadaran quinazolinone kuma yana nuna halaye na musamman na kimiyyar sinadarai wanda hakan ya sa ya zama mai amfani ga kokarin gano magunguna da nazarin dangantaka tsakanin tsari da aiki wajen samar da sabbin magunguna masu warkarwa.
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5,6-Difluoro-2,3-dihydro-1H-isoindol-1-one CAS:1192040-50-8
5,6-Difluoro-2,3-dihydro-1H-isoindol-1-one, wanda aka san shi da halaye masu yawa, yana aiki a matsayin babban mahaɗi a fannoni daban-daban na bincike da masana'antu. Tare da dabarar sinadarai ta C8H6F2NO, yana da wani muhimmin tushen isoindolone wanda aka maye gurbinsa da ƙwayoyin fluorine guda biyu, yana ba da halaye daban-daban ga tsarinsa. Wannan mahaɗin yana samun aikace-aikace a fannoni daban-daban saboda bambancin amsawarsa da yuwuwar haɗa ƙwayoyin hadaddun tare da mahimmancin kimiyyar magunguna da kayan aiki.
