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Sitagliptin Phosphate CAS:654671-78-0 Mai Kaya na Masana'anta

Sitagliptin Phosphateshine sabon maganin dipeptidyl peptidase IV na farko daga Merck don maganin ciwon suga na nau'in 2 ba tare da ƙara nauyi ba kuma yawan hypoglycemia yayi kama da placebo. Sitagliptin yana aiki ta hanyar inganta tsarin incretin na jiki, wanda ke taimakawa wajen daidaita glucose ta hanyar shafar ƙwayoyin β da α a cikin pancreas.


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Sitagliptin Phosphate wani maganin hana ciwon suga ne na trizolopyrazine dipeptidyl peptidase IV. An amince da Sitagliptin kwanan nan don maganin ciwon suga na nau'in II. Sitagliptin phosphate wani nau'in maganin hana ciwon suga ne na dipeptidyl peptidase Ⅳ(DDP-4) wanda kamfanin Jamus Merck ya ƙirƙiro kuma da farko ya sami amincewar Hukumar Abinci da Magunguna ta Amurka don maganin ciwon suga na nau'in 2, sabon magani ne na hana ciwon suga, wanda zai iya inganta ikon jiki na rage yawan glucose a jini, da kuma ƙaruwar incretin ta halitta ta hanyar hana aikin wannan enzyme, gami da matakan glucagon-like peptide 1 da insulinotropic peptide wanda ke dogara da glucose, wanda hakan ke haifar da pancreas don inganta samar da insulin da kuma dakatar da samar da glucose a hanta, da kuma rage tasirin asibiti na yawan glucose a jini.

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shafi 365 (1)

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shafi 338 (1)

Ƙarin Bayani:

Tsarin aiki C16H15F6N5O.H3PO4
Gwaji 99%
Bayyanar Foda fari zuwa farin da ba a kashe ba
Lambar CAS 654671-78-0
shiryawa 25KG
Rayuwar shiryayye Shekaru 2
Ajiya A adana a wuri mai sanyi da bushewa
Takardar shaida ISO.

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