Bel da Hanya: Haɗin gwiwa, Jituwa da Cin Nasara
samfurori

Kayayyaki

Mirabegron CAS:223673-61-8 Mai Kaya na Masana'anta

Ana amfani da Mirabegron don magance gaggawa, yawan fitsari, da kuma rashin isasshen fitsari da ke tattare da mafitsara mai aiki fiye da kima (OAB). Ana haɗa Mirabegron ta hanyar haɗa 4-nitrophenethyl amine zuwa (R)-2-hydroxy-2-phenylacetic acid. Ana rage amide ɗin da ke fitowa zuwa amine. Daga nan sai a rage rukunin nitro kuma a haɗa sakamakon zuwa 2-(2-aminothiazol-4-yl) acetic acid don samar da mirabegron.


Cikakken Bayani game da Samfurin

Alamun Samfura

Aikace-aikace da Tasiri

Mirabegron wani agonist ne mai aiki da baki na β3-adrenoceptor wanda Astellas Pharma ke samarwa don maganin mafitsara mai aiki fiye da kima (OAB). Maganin wani antagonist ne nanomolar EC50 akan gwajin biochemical na β3-AR na ɗan adam tare da kyakkyawan zaɓi fiye da b1- da β2-ARs. Mirabegron ya nuna sabon tsari ta hanyar niyya ga β3-AR don shakatawa mafitsara don taimakawa wajen magance alamun OAB kamar ƙaruwar gaggawar fitsari da yawan fitsari da kuma rashin isasshen ruwa cikin gaggawa. Duk da haka, mirabegron wani antagonist ne na cytochrome P450 2D6, kuma yana haifar da damuwa game da hulɗar magunguna da magunguna tare da shan wasu abubuwan cytochrome P450 2D6 tare da lokaci guda.

Samfurin Samfuri

图片272(1)
图片273(1)

Shirya Samfurin:

图片210(1)

Ƙarin Bayani:

Tsarin aiki C21H24N4O2S
Gwaji 99%
Bayyanar Foda fari zuwa rawaya mai haske
Lambar CAS 223673-61-8
shiryawa 25KG
Rayuwar shiryayye Shekaru 2
Ajiya A adana a wuri mai sanyi da bushewa
Takardar shaida ISO.

  • Na baya:
  • Na gaba:

  • Rubuta saƙonka a nan ka aika mana da shi