Mirabegron CAS:223673-61-8 Mai Kaya na Masana'anta
Mirabegron wani agonist ne mai aiki da baki na β3-adrenoceptor wanda Astellas Pharma ke samarwa don maganin mafitsara mai aiki fiye da kima (OAB). Maganin wani antagonist ne nanomolar EC50 akan gwajin biochemical na β3-AR na ɗan adam tare da kyakkyawan zaɓi fiye da b1- da β2-ARs. Mirabegron ya nuna sabon tsari ta hanyar niyya ga β3-AR don shakatawa mafitsara don taimakawa wajen magance alamun OAB kamar ƙaruwar gaggawar fitsari da yawan fitsari da kuma rashin isasshen ruwa cikin gaggawa. Duk da haka, mirabegron wani antagonist ne na cytochrome P450 2D6, kuma yana haifar da damuwa game da hulɗar magunguna da magunguna tare da shan wasu abubuwan cytochrome P450 2D6 tare da lokaci guda.
| Tsarin aiki | C21H24N4O2S |
| Gwaji | 99% |
| Bayyanar | Foda fari zuwa rawaya mai haske |
| Lambar CAS | 223673-61-8 |
| shiryawa | 25KG |
| Rayuwar shiryayye | Shekaru 2 |
| Ajiya | A adana a wuri mai sanyi da bushewa |
| Takardar shaida | ISO. |
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